KISS1R Signaling
Kisspeptins are endogenous ligands of the kisspeptin receptor KISS1R, historically known as GPR54. Foundational receptor studies characterized kisspeptin-mediated signaling in receptor-expressing experimental systems, including phospholipase-C-associated signaling, intracellular calcium mobilization and downstream kinase pathways. KP-10 contains the conserved C-terminal sequence required for kisspeptin receptor activity and is widely used as a research ligand for investigating KISS1R signaling.



